Názov: Structure-based discovery of the first allosteric inhibitors of cyclin-dependent kinase 2 : [Štruktúra na báze objavov prvých alosterických inhibítorov cyklin-dependentné kinázy 2]
Zápis: RASTELLI, Giulio - ANIGHORO, Andrew - CHRIPKOVÁ, Martina - CARRASSA, Laura - BROGGINI, Massimo. Structure-based discovery of the first allosteric inhibitors of cyclin-dependent kinase 2 : [Štruktúra na báze objavov prvých alosterických inhibítorov cyklin-dependentné kinázy 2] In: Cell Cycle. 2014. ISSN 1538-4101, Vol. 13, č. 14(2014), s. 2296-2305.
(2014: 5.006 - IF, 141 - H-index, 0.914 - IF 5y, 2.048 - SJR, Q1 - SJR Best Q, Q2 - JCR Best Q)
Rok vydania: 2014
Kategória: ADC - Vedecké práce v zahraničných karentovaných časopisoch
Autori:RASTELLI Giulio40 %
ANIGHORO Andrew15 %
CHRIPKOVÁ Martina15 %
CARRASSA Laura10 %
BROGGINI Massimo20 %
Vydanie: Cell Cycle
Vol. 13, č. 14(2014), s. 2296-2305
Krajina vydania: Slovensko
ISSN:1538-4101
Oblasť výskumu: 180 - Lekárske, farmaceutické a nelekárske zdravotnícke vedy
Scientometria: 2014: 5.006 - IF, 141 - H-index, 0.914 - IF 5y, 2.048 - SJR, Q1 - SJR Best Q, Q2 - JCR Best Q
Jazyk: anglický
URL na ARL: https://arl4.library.sk/arl-uvlk/sk/detail-uvlk_un_cat-0021935-Structurebased-discovery-of-the-first-allosteric-inhibitors-of-cyclindependent-kinase-2/
Ohlasy:
2018: [1] CRAVEN, Gregory B. - AFFRON, Dominic P. - ALLEN, Charlotte E. - MATTHIES, Stefan - GREENER, Joe G. - MORGAN, Rhodri M. L. - TATE, Edward W. - ARMSTRONG, Alan - MANN, David J. High-Throughput Kinetic Analysis for Target-Directed Covalent Ligand Discovery. In ANGEWANDTE CHEMIE-INTERNATIONAL EDITION. ISSN 1433-7851, 2018, vol. 57, no. 19, pp. 5257-5261. [WoS]
2017: [1] BAJUSZ, David - FERENCZY, Gyorgy G. - KESERU, Gyorgy M. Structure-based Virtual Screening Approaches in Kinase-directed Drug Discovery. In CURRENT TOPICS IN MEDICINAL CHEMISTRY. ISSN 1568-0266, 2017, vol. 17, no. 20, pp. 2235-2259. [WoS]
2017: [1] BEHERA, Pabitra Mohan - DIXIT, Anshuman. The story of kinase inhibitors development with special reference to allosteric site. In Drug Design: Principles and Applications, 2017-08-09, pp. 57-68. [Scopus]
2017: [1] GREENER, Joe G. - FILIPPIS, Ioannis - STERNBERG, Michael J. E. Predicting Protein Dynamics and Allostery Using Multi-Protein Atomic Distance Constraints. In STRUCTURE. ISSN 0969-2126, 2017, vol. 25, no. 3, pp. 546-558. [WoS]
2017: [1] KALRA, Sourav - JOSHI, Gaurav - MUNSHI, Anjana - KUMAR, Raj. Structural insights of cyclin dependent kinases: Implications in design of selective inhibitors. In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234, 2017, vol. 142, no., pp. 424-458. [WoS]
2017: [1] PELLERANO, Morgan - TCHERNIUK, Sergey - PERALS, Corine - THI NHU NGOC VAN - GARCIN, Elsa D. - MAHUTEAU-BETZER, Florence - TEULADE-FICHOU, Marie-Paule - MORRIS, May C. Targeting Conformational Activation of CDK2 Kinase. In BIOTECHNOLOGY JOURNAL. ISSN 1860-6768, 2017, vol. 12, no. 8, pp. [WoS]
2017: [1] TUTONE, Marco - ALMERICO, Anna Maria. Recent advances on CDK inhibitors: An insight by means of in silico methods. In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234, 2017, vol. 142, no., pp. 300-315. [WoS]
2017: [1] WANG, Huiwen - WANG, Kaili - GUAN, Zeyu - JIAN, Yiren - JIA, Ya - KASHANCHI, Fatah - ZENG, Chen - ZHAO, Yunjie. Computational study of non-catalytic T-loop pocket on CDK proteins for drug development. In CHINESE PHYSICS B. ISSN 1674-1056, 2017, vol. 26, no. 12, pp. [WoS]
2016: [1] CAPORUSCIO, Fabiana - RASTELLI, Giulio. Exploiting computationally derived out-of-the-box protein conformations for drug design. In Future Medicinal Chemistry. ISSN 17568919, 2016-10-01, 8, 15, pp. 1887-1897. [Scopus]
2016: [1] CARLINO, Luca - RASTELLI, Giulio. Dual Kinase-Bromodomain Inhibitors in Anticancer Drug Discovery: A Structural and Pharmacological Perspective. In Journal of Medicinal Chemistry. ISSN 00222623, 2016-10-27, 59, 20, pp. 9305-9320. [Scopus]
2016: [1] CHILÀ, Rosaria - GUFFANTI, Federica - DAMIA, Giovanna. Role and therapeutic potential of CDK12 in human cancers. In Cancer Treatment Reviews. ISSN 03057372, 2016-11-01, 50, pp. 83-88. [Scopus]
2016: [1] LI, Tinghan - WENG, Tianwei - ZUO, Minzan - WEI, Zhihui - CHEN, Ming - LI, Zhiyu. Recent progress of cyclin-dependent kinase inhibitors as potential anticancer agents. In Future Medicinal Chemistry. ISSN 17568919, 2016-11-01, 8, 17, pp. 2047-2076. [Scopus]
2016: [1] LU, Fang - LUO, Ganggang - QIAO, Liansheng - JIANG, Ludi - LI, Gongyu - ZHANG, Yanling. Virtual screening for potential allosteric inhibitors of cyclin-dependent kinase 2 from traditional chinese medicine. In Molecules, 2016-09-01, 21, 9, pp. [Scopus]
2015: [1] LI, Yan - ZHANG, Jingxiao - GAO, Weimin - ZHANG, Lilei - PAN, Yanqiu - ZHANG, Shuwei - WANG, Yonghua. Insights on Structural Characteristics and Ligand Binding Mechanisms of CDK2. In INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES. ISSN 1422-0067, 2015, vol. 16, no. 5, pp. 9314. [WoS]
2015: [1] SANCHEZ-MARTINEZ, Concepcion - GELBERT, Lawrence M. - JOSE LALLENA, Maria - DE DIOS, Alfonso. Cyclin dependent kinase (CDK) inhibitors as anticancer drugs. In BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. ISSN 0960-894X, 2015, vol. 25, no. 17, pp. 3420. [WoS]
2015: [1] WU, Peng - CLAUSEN, Mads H. - NIELSEN, Thomas E. Allosteric small-molecule kinase inhibitors. In PHARMACOLOGY & THERAPEUTICS. ISSN 0163-7258, 2015, vol. 156, no., pp. 59. [WoS]
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